SCHEMBL6879909

SCHEMBL6879909

OC/C=C(/F)c1ccc(-c2ccncc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
KIF11 P52732 2/20 0.39
CYP17A1 P05093 1/20 0.38
PRKACA P17612 6/20 0.37
PRKX P51817 6/20 0.37
ROCK1 Q13464 6/20 0.37
CLK4 Q9HAZ1 6/20 0.37
ROCK2 O75116 5/20 0.37
PRKG1 Q13976 5/20 0.37
PKN2 Q16513 5/20 0.37
GSK3A P49840 5/20 0.37
GSK3B P49841 5/20 0.37
RPS6KB1 P23443 4/20 0.37
PRKG2 Q13237 4/20 0.37
RPS6KA5 O75582 4/20 0.37
MAPK1 P28482 4/20 0.37
SGK2 Q9HBY8 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6879912 1.00 HDAC1 (0.42) HDAC1HDAC6MAPTLMNAKIF11
SCHEMBL6879903 1.00 HDAC1 (0.42) HDAC1HDAC6MAPTLMNAKIF11
SCHEMBL6877827 0.82 ATM (0.39) HDAC1MAP4K4ERN1
SCHEMBL6877820 0.82 ATM (0.39) HDAC1MAP4K4ERN1
SCHEMBL6877823 0.82 ATM (0.39) HDAC1MAP4K4ERN1
SCHEMBL6877224 0.82 MKNK1 (0.54) MAPTLMNAKIF11SMN1; SMN2
SCHEMBL6877227 0.82 MKNK1 (0.54) MAPTLMNAKIF11SMN1; SMN2
SCHEMBL6877229 0.82 MKNK1 (0.54) MAPTLMNAKIF11SMN1; SMN2
SCHEMBL6878376 0.80 CYP2D6 (0.43) MAPTPRKACAPRKXROCK1CLK4
SCHEMBL6878371 0.80 CYP2D6 (0.43) MAPTPRKACAPRKXROCK1CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6825170-B2 ERYTHROMYCIN TYPE MACROLIDE WITH A FUSED OXAZOLONE RING ORTHO-MCNEIL PHARMACEUTICAL, INC. 2004-11-30 US disclosed