SCHEMBL6878418

SCHEMBL6878418

COc1ccc2[nH]cc(CNCC3CCC(Nc4cc(N(C)C)c5ccccc5n4)CC3)c2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.44
CYP1A2 P05177 6/20 0.44
CYP3A4 P08684 6/20 0.44
CYP2D6 P10635 6/20 0.44
CYP2C19 P33261 6/20 0.44
LMNA P02545 5/20 0.44
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
CYP2C9 P11712 4/20 0.44
ALOX15 P16050 4/20 0.44
USP2 O75604 4/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 3/20 0.44
CLK4 Q9HAZ1 3/20 0.44
TSHR P16473 2/20 0.44
CASP1 P29466 1/20 0.44
RECQL P46063 1/20 0.44
BLM P54132 1/20 0.44
CASP7 P55210 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6878414 1.00 TP53 (0.44) TP53CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6876199 0.90 MCHR1 (0.47) TP53CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6876191 0.90 MCHR1 (0.47) TP53CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6873072 0.90 MCHR1 (0.45) TP53LMNAMEN1KMT2AUSP2
SCHEMBL6873067 0.90 MCHR1 (0.45) TP53LMNAMEN1KMT2AUSP2
SCHEMBL6466930 0.89 MCHR1 (0.49) LMNASIGMAR1KDM4ESMN1; SMN2MCHR1
SCHEMBL6875524 0.89 MCHR1 (0.49) LMNASIGMAR1KDM4ESMN1; SMN2MCHR1
SCHEMBL6873885 0.86 MCHR1 (0.46) TP53CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL6873877 0.86 MCHR1 (0.46) TP53CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL13793582 0.86 MCHR1 (0.57) TP53CYP1A2CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed