SCHEMBL6879063

SCHEMBL6879063

CCOC(=O)c1cccc(NC(=O)NC2CCC(Nc3cc(N(C)C)c4ccccc4n3)CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.49
CSNK2A1 P68400 1/20 0.49
MAPT P10636 7/20 0.49
TP53 P04637 4/20 0.49
MAPK1 P28482 2/20 0.46
TSHR P16473 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 2/20 0.45
ALDH1A1 P00352 2/20 0.45
RAB9A P51151 2/20 0.45
CCKBR P32239 1/20 0.45
MEN1 O00255 1/20 0.45
ABCB1 P08183 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
NAMPT P43490 1/20 0.44
THRB P10828 1/20 0.44
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6879057 1.00 GSK3B (0.49) GSK3BCSNK2A1MAPTTP53MAPK1
SCHEMBL6869115 0.92 MAPT (0.48) MAPTTP53MAPK1TSHRSMN1; SMN2
SCHEMBL6869121 0.92 MAPT (0.48) MAPTTP53MAPK1TSHRSMN1; SMN2
SCHEMBL4036980 0.85 MCHR1 (0.62) GSK3BCSNK2A1MAPTTP53NPC1
SCHEMBL4036978 0.85 MCHR1 (0.62) GSK3BCSNK2A1MAPTTP53NPC1
SCHEMBL6872848 0.83 NPC1 (0.46) MAPTNPC1ALDH1A1RAB9AMEN1
SCHEMBL6872842 0.83 NPC1 (0.46) MAPTNPC1ALDH1A1RAB9AMEN1
SCHEMBL6457991 0.81 EPHX1 (0.47) TP53SMN1; SMN2KMT2ALMNA
SCHEMBL6457984 0.81 EPHX1 (0.47) TP53SMN1; SMN2KMT2ALMNA
SCHEMBL6877850 0.81 EPHX1 (0.49) TP53SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed