SCHEMBL6879976

SCHEMBL6879976

O=C(OCc1ccccc1)N1CC2(CCNCC2)c2ccc(Br)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.47
BIRC2 Q13490 1/20 0.47
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
GAA P10253 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
HTR2C P28335 1/20 0.39
CASP1 P29466 1/20 0.37
TACR1 P25103 2/20 0.36
P2RX4 Q99571 2/20 0.36
ENPP2 Q13822 1/20 0.36
ATXN2 Q99700 1/20 0.36
P2RY1 P47900 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6544398 0.87 NPC1 (0.51) XIAPBIRC2HDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL7565105 0.86 NPC1 (0.50) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL7542146 0.81 NPC1 (0.43) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL6887035 0.81 NPC1 (0.47) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL15771793 0.76 NPC1 (0.39) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL15772117 0.76 NPC1 (0.39) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL14295982 0.75 HDAC1 (0.54) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL6879988 0.74 XIAP (0.42) XIAPBIRC2HDAC1HDAC8HDAC6
SCHEMBL6543487 0.74 NOTUM (0.55) HDAC1HDAC6GAASMN1; SMN2P2RY1
SCHEMBL1670307 0.73 NPC1 (0.54) XIAPBIRC2HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377293-A1 ARYL AND BIARYL PIPERIDINES USED AS MCH ANTAGONISTS PHARMACOPEIA, INC. (US) 2004-01-07 EP disclosed
WO-2002083134-A1 ARYL AND BIARYL PIPERIDINES USED AS MCH ANTAGONISTS PHARMACOPEIA, INC. (US) 2002-10-24 WO disclosed