SCHEMBL6887035

SCHEMBL6887035

O=C(OCc1ccccc1)N1CC2(CCNCC2)c2c(Br)cccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HTR2C P28335 1/20 0.40
P2RX4 Q99571 2/20 0.40
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
P2RX1 P51575 1/20 0.39
P2RX3 P56373 1/20 0.39
CTRB1 P17538 1/20 0.38
TACR1 P25103 1/20 0.38
XIAP P98170 1/20 0.37
BIRC2 Q13490 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6544398 0.84 NPC1 (0.51) NPC1RAB9ASMN1; SMN2GAAMAPK1
Hydrochloric Acid SCHEMBL7565105 0.83 NPC1 (0.50) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL6879976 0.81 XIAP (0.47) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL7542146 0.77 NPC1 (0.43) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL17134660 0.76 NPC1 (0.56) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL3668093 0.74 TSHR (0.43) HDAC1HDAC8HDAC6DDB1CRBN
SCHEMBL15561394 0.74 PTGDR2 (0.40) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL30659272 0.72 NPC1 (0.46) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL15561354 0.72 XDH (0.39) NPC1RAB9ASMN1; SMN2GAAMAPK1
SCHEMBL19439193 0.72 NPC1 (0.67) NPC1RAB9ASMN1; SMN2GAAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377293-A1 ARYL AND BIARYL PIPERIDINES USED AS MCH ANTAGONISTS PHARMACOPEIA, INC. (US) 2004-01-07 EP disclosed
WO-2002083134-A1 ARYL AND BIARYL PIPERIDINES USED AS MCH ANTAGONISTS PHARMACOPEIA, INC. (US) 2002-10-24 WO disclosed