SCHEMBL6880487

SCHEMBL6880487

COc1ccc(NC(=O)N[C@H]2CC[C@@H](Nc3nc4c(c(N(C)C)n3)CCCC4)CC2)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.45
ALDH1A1 P00352 3/20 0.45
HPGD P15428 1/20 0.45
MAPT P10636 3/20 0.44
LMNA P02545 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
MALT1 Q9UDY8 6/20 0.44
NPC1 O15118 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
EPHX2 P34913 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ADRA2A P08913 2/20 0.41
MCHR1 Q99705 2/20 0.41
BCL6 P41182 1/20 0.40
DUSP3 P51452 1/20 0.40
PTPN5 P54829 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6880492 1.00 TP53 (0.45) TP53ALDH1A1HPGDMAPTLMNA
SCHEMBL6458641 0.92 SMN1; SMN2 (0.47) TP53ALDH1A1MAPTLMNANPSR1
SCHEMBL6458645 0.92 SMN1; SMN2 (0.47) TP53ALDH1A1MAPTLMNANPSR1
SCHEMBL6867531 0.90 MCHR1 (0.49) ALDH1A1MAPTNPC1TSHRHTT
SCHEMBL6867526 0.90 MCHR1 (0.49) ALDH1A1MAPTNPC1TSHRHTT
SCHEMBL6873496 0.90 NPC1 (0.57) ALDH1A1NPC1TSHRHTTRAB9A
SCHEMBL6873499 0.90 NPC1 (0.57) ALDH1A1NPC1TSHRHTTRAB9A
SCHEMBL6878062 0.88 MEN1 (0.58) ALDH1A1MAPTLMNANPC1TSHR
SCHEMBL6872085 0.88 KMT2A (0.43) TP53ALDH1A1MAPTLMNATSHR
SCHEMBL6878058 0.88 MEN1 (0.58) ALDH1A1MAPTLMNANPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1464335-A2 Quinoline, tetrahydroquinoline and pyrimidine derivatives as mch antagonist Taisho Pharmaceutical Co. Ltd. (JP) 2004-10-06 EP disclosed