SCHEMBL6880652

SCHEMBL6880652

O=C(Cc1csc(NC(=O)OCC23CC4CC(CC2C4)C3)n1)NO

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 17/20 0.47
PDE1A P54750 7/20 0.47
PDE1B Q01064 7/20 0.47
PDE1C Q14123 7/20 0.47
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758918 0.81 PDE5A (0.44) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1759205 0.78 CNR2 (0.62) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL6876782 0.78 PDE5A (0.42) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL6878810 0.78 PDE5A (0.39) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758713 0.77 PDE5A (0.54) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758738 0.77 PDE5A (0.48) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758649 0.76 EPHX2 (0.63) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL6880659 0.76 PDE5A (0.47) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL6880557 0.74 TSHR (0.44) PDE5APDE1APDE1BPDE1CKDM4E
SCHEMBL1758935 0.74 PDE5A (0.39) PDE5APDE1APDE1BPDE1CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed