SCHEMBL1759205

SCHEMBL1759205

O=C(Cc1csc(NC(=O)C23CC4CC(CC(C4)C2)C3)n1)NO

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.62
GAA P10253 1/20 0.61
HTT P42858 1/20 0.61
PDE5A O76074 16/20 0.53
KDM4E B2RXH2 2/20 0.53
PDE1A P54750 6/20 0.51
PDE1B Q01064 6/20 0.51
PDE1C Q14123 6/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1759195 0.92 GAA (0.53) CNR2GAAHTTPDE5AKDM4E
SCHEMBL1758713 0.84 PDE5A (0.54) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758649 0.83 EPHX2 (0.63) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758692 0.79 PDE5A (0.56) GAAHTTPDE5AKDM4EPDE1A
SCHEMBL6880652 0.78 PDE5A (0.47) GAAHTTPDE5AKDM4EPDE1A
SCHEMBL3607475 0.76 PDE5A (0.70) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL962008 0.74 CNR2 (0.67) CNR2GAAHTTKDM4E
SCHEMBL6879293 0.74 GAA (0.49) CNR2GAAHTT
SCHEMBL1758655 0.74 CNR2 (0.59) CNR2GAAHTTKDM4E
SCHEMBL1758930 0.74 PDE5A (0.49) PDE5AKDM4EPDE1APDE1BPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO claimed