SCHEMBL6880838

SCHEMBL6880838

CC(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCCCNC(=O)C(F)(F)F)C(=O)Nc1ccc2ccc(=O)oc2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
NPBWR1 P48145 1/20 0.36
MAP2K1 Q02750 1/20 0.34
FPR2 P25090 1/20 0.34
PGR P06401 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CAPN1 P07384 1/20 0.34
NPY4R P50391 1/20 0.34
KMT2A Q03164 1/20 0.33
CA9 Q16790 1/20 0.33
ACHE P22303 1/20 0.33
CA4 P22748 1/20 0.33
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11906012 0.90 CA9 (0.46) CA1ALDH1A1KDM4EMAP2K1SMN1; SMN2
SCHEMBL6877904 0.90 CA9 (0.46) CA1ALDH1A1KDM4EMAP2K1SMN1; SMN2
SCHEMBL11983772 0.81 CA12 (0.50) CA1ALDH1A1KDM4ESMN1; SMN2L3MBTL1
SCHEMBL10315740 0.81 CA12 (0.50) CA1ALDH1A1KDM4ESMN1; SMN2L3MBTL1
SCHEMBL10315741 0.77 CA12 (0.50) CA1ALDH1A1KDM4ESMN1; SMN2MAPT
SCHEMBL11983774 0.77 CA12 (0.50) CA1ALDH1A1KDM4ESMN1; SMN2MAPT
SCHEMBL18220762 0.74 CA12 (0.44) CA1ALDH1A1KDM4ESMN1; SMN2NPY4R
SCHEMBL3098313 0.73 KDM4E (0.49) CA1ALDH1A1KDM4ESMN1; SMN2KMT2A
SCHEMBL18220760 0.73 CA1 (0.47) SIRT5CA1CA2ALDH1A1KDM4E
SCHEMBL16234039 0.71 CACNA1B (0.41) CA2ALDH1A1NPBWR1SMN1; SMN2CAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084991-A2 FLUORINATED HDAC INHIBITORS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-07-14 WO disclosed