SCHEMBL6880856

SCHEMBL6880856

Nc1cnn2cc(C#Cc3ccccc3)cnc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMPD3 Q9NY59 1/20 0.44
GRM5 P41594 8/20 0.43
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
APP P05067 1/20 0.38
GRM4 Q14833 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1992762 0.79 CDK2 (0.49) GRM5MAPTKDM4EMEN1NPC1
SCHEMBL31470548 0.77 SMPD3 (0.44) SMPD3KDM4EMEN1NPC1ALDH1A1
SCHEMBL1991466 0.72 KIT (0.51) GRM5
SCHEMBL1996090 0.72 GRM5 (0.44) GRM5MEN1NPC1KMT2AADORA2A
SCHEMBL4395064 0.70 SMPD3 (0.52) SMPD3KDR
SCHEMBL403731 0.68 GRM5 (0.61) GRM5MAPTKDM4EMEN1NPC1
SCHEMBL22834525 0.67 SMPD3 (0.48) SMPD3KDR
SCHEMBL21893829 0.67 SMPD3 (0.48) SMPD3KDR
Hydrochloric Acid SCHEMBL22835004 0.66 SMPD3 (0.47) SMPD3KDR
Hydrochloric Acid SCHEMBL22834582 0.66 SMPD3 (0.47) SMPD3MAPTKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073172-A1 ETHYNYL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed