SCHEMBL688196

SCHEMBL688196

O=C(O)C[C@@H](Cc1cccc(C(F)(F)F)c1)NC(=O)Nc1c(O)ccn(Cc2ccccc2Cl)c1=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.47
MAPT P10636 4/20 0.44
THRB P10828 1/20 0.44
PTGER3 P43115 8/20 0.42
CYP1A2 P05177 1/20 0.42
FFAR2 O15552 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPK1 P28482 1/20 0.41
MME P08473 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
LMNA P02545 2/20 0.39
TP53 P04637 2/20 0.38
RXFP1 Q9HBX9 1/20 0.38
ATM Q13315 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687905 0.86 PTGER3 (0.46) MAPTTHRBPTGER3CYP1A2KDM4E
SCHEMBL27741944 0.86 CTSA (0.47) MAPTTHRBPTGER3KDM4EALDH1A1
SCHEMBL687768 0.86 CTSA (0.47) MAPTTHRBPTGER3KDM4EALDH1A1
SCHEMBL687685 0.84 PTGER3 (0.48) MAPTPTGER3CYP1A2KDM4EALDH1A1
SCHEMBL688064 0.84 PTGER3 (0.48) MAPTPTGER3CYP1A2KDM4EALDH1A1
SCHEMBL688237 0.84 KDM4E (0.46) PTGER3CYP1A2KDM4EALDH1A1SMN1; SMN2
SCHEMBL687702 0.83 MAPT (0.50) MAPTTHRBPTGER3CYP1A2KDM4E
SCHEMBL688152 0.83 LCK (0.42) PTGER3KDM4EALDH1A1SMN1; SMN2MAPK1
SCHEMBL687900 0.82 PTGER3 (0.48) PTGER3CYP1A2KDM4EALDH1A1SMN1; SMN2
SCHEMBL687043 0.82 CTSA (0.45) MAPTTHRBPTGER3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed