SCHEMBL688215

SCHEMBL688215

COc1ccccc1-c1cccc([C@H](CC(=O)O)NC(=O)Nc2c(O)c(C)cn(Cc3ccccc3Cl)c2=O)c1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGER3 P43115 4/20 0.43
CTSA P10619 7/20 0.41
ITGB1 P05556 3/20 0.40
ITGA4 P13612 3/20 0.40
MAPT P10636 1/20 0.37
P2RX7 Q99572 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688669 0.92 PTGER3 (0.42) PTGER3CTSAITGB1ITGA4MAPT
SCHEMBL688474 0.92 PTGER3 (0.39) PTGER3CTSAITGB1ITGA4
SCHEMBL687228 0.90 GNRHR (0.39) PTGER3CTSAITGB1ITGA4
SCHEMBL686799 0.89 PTGER3 (0.51) PTGER3CTSAMAPT
SCHEMBL688233 0.88 PTGER3 (0.43) PTGER3CTSAMAPTP2RX7
SCHEMBL688379 0.88 PTGER3 (0.42) PTGER3CTSA
SCHEMBL688343 0.88 PTGER3 (0.43) PTGER3CTSAMAPTP2RX7
SCHEMBL687991 0.88 GNRHR (0.38) PTGER3CTSAITGB1ITGA4
SCHEMBL687527 0.88 ITGB1 (0.42) PTGER3CTSAITGB1ITGA4MAPT
SCHEMBL688878 0.88 PTGER3 (0.41) PTGER3CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed