SCHEMBL6882889

SCHEMBL6882889

Cc1c(-c2ccnn2-c2ccc(N)cc2)cc(C(=O)NCCC[N+]2(C)CCCC2)c(=O)n1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.59
NPSR1 Q6W5P4 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CCR1 P32246 4/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MAPT P10636 2/20 0.38
HSP90AA1 P07900 1/20 0.38
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
HTR2A P28223 3/20 0.36
HTR2C P28335 3/20 0.36
SLC6A4 P31645 2/20 0.36
LMNA P02545 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1604972 0.91 ELANE (0.73) ELANENPSR1KDM4E
Iodide SCHEMBL1603664 0.91 ELANE (0.72) ELANE
SCHEMBL1604115 0.89 ELANE (0.72) ELANENPSR1KDM4E
Acetic Acid SCHEMBL1603917 0.87 ELANE (0.69) ELANECCR1
SCHEMBL1604046 0.87 ELANE (0.75) ELANENPSR1KDM4ECCR1MEN1
SCHEMBL6882229 0.86 ELANE (0.65) ELANENPSR1KDM4ECCR1MEN1
Acetic Acid SCHEMBL1604007 0.85 ELANE (0.72) ELANENPSR1KDM4ECCR1
SCHEMBL8219783 0.84 ELANE (0.66) ELANENPSR1KDM4ECCR1MEN1
SCHEMBL14922185 0.80 ELANE (0.81) ELANENPSR1KDM4ECCR1MEN1
SCHEMBL1604014 0.80 ELANE (0.74) ELANEHTR2AHTR2CSLC6A4ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011039528-A1 2-PYRIDONE COMPOUNDS USED AS INHIBITORS OF NEUTROPHIL ELASTASE ASTRAZENECA AB (SE) 2011-04-07 WO disclosed