SCHEMBL6883374

SCHEMBL6883374

O=c1[nH]c2ccc(Br)cc2c(OCC2CC=CC=N2)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.44
ALDH1A1 P00352 4/20 0.41
MAPT P10636 3/20 0.41
TSHR P16473 1/20 0.41
CASP7 P55210 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GRIN2D O15399 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
POLB P06746 1/20 0.38
PADI4 Q9UM07 2/20 0.37
IKBKB O14920 1/20 0.36
CHUK O15111 1/20 0.36
AKT1 P31749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2680869 0.78 PDE2A (0.57) PDE2AALDH1A1MAPTTSHRCASP7
SCHEMBL936269 0.75 HDAC1 (0.50) PDE2AALDH1A1MAPTTSHRCASP7
SCHEMBL6883842 0.74 PDE2A (0.61) PDE2AGRIN2DGRIN2AGRIN2BGRIN2C
SCHEMBL936355 0.73 PDE2A (0.57) PDE2AALDH1A1MAPTTSHRCASP7
SCHEMBL15648185 0.66 KDM4E (0.70) ALDH1A1MAPTTSHRCASP7HSD17B10
SCHEMBL24095578 0.66 MEN1 (0.59) ALDH1A1MAPTTSHRCASP7HSD17B10
SCHEMBL31384364 0.66 ALDH1A1 (0.63) ALDH1A1MAPTTSHRCASP7HSD17B10
SCHEMBL25849925 0.64 MEN1 (0.63) ALDH1A1MAPTTSHRCASP7HSD17B10
SCHEMBL935454 0.64 PDE2A (0.80) PDE2AGRIN2DGRIN2AGRIN2BGRIN2C
SCHEMBL962565 0.62 PDE2A (0.77) PDE2AALDH1A1MAPTTSHRCASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011312-A1 QUINOLINONE PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-01-27 WO disclosed