SCHEMBL6885264

SCHEMBL6885264

CC(C)(O)C#Cc1ccc2[nH]c(=O)c(C3CC=CS3)c(OCC3CCOCC3)c2c1

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 4/20 0.65
CYP2D6 P10635 3/20 0.33
PIKFYVE Q9Y2I7 4/20 0.32
MAP3K14 Q99558 4/20 0.32
TTBK1 Q5TCY1 2/20 0.32
PAK4 O96013 1/20 0.32
PRKX P51817 1/20 0.32
TAOK1 Q7L7X3 1/20 0.32
TSSK3 Q96PN8 1/20 0.32
TSSK1B Q9BXA7 1/20 0.32
TAOK3 Q9H2K8 1/20 0.32
PAK6 Q9NQU5 1/20 0.32
PAK5 Q9P286 1/20 0.32
TAOK2 Q9UL54 1/20 0.32
IDH1 O75874 1/20 0.31
ACACB O00763 1/20 0.31
CHUK O15111 1/20 0.30
PDE9A O76083 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885522 0.82 PDE2A (0.45) PDE2ACYP2D6PDE9A
SCHEMBL957022 0.79 PDE2A (1.00) PDE2ACYP2D6PIKFYVEMAP3K14TTBK1
SCHEMBL2680484 0.70 PDE2A (0.85) PDE2APIKFYVEMAP3K14TTBK1PAK4
SCHEMBL6346581 0.65 PDE2A (0.53) PDE2ACYP2D6IDH1
SCHEMBL6345622 0.64 PDE2A (0.75) PDE2ACYP2D6
SCHEMBL962565 0.58 PDE2A (0.77) PDE2ACYP2D6PDE9A
SCHEMBL2680415 0.58 PDE2A (0.66) PDE2APIKFYVEMAP3K14TTBK1PAK4
Propionic Acid SCHEMBL4162291 0.56 PDE2A (0.39) PDE2APIKFYVEMAP3K14TTBK1PAK4
SCHEMBL9214507 0.56 ACACB (0.50) ACACB
SCHEMBL6349695 0.56 PDE2A (0.52) PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011312-A1 QUINOLINONE PDE2 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-01-27 WO disclosed