SCHEMBL6885276

SCHEMBL6885276

COCC1CCCN1C(=O)c1cc(N)c2nc(-c3ccc(C)o3)nn2c1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.83
ADORA1 P30542 2/20 0.49
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12923691 1.00 ADORA2A (0.83) ADORA2AADORA1NPC1RAB9A
SCHEMBL22722588 1.00 ADORA2A (0.83) ADORA2AADORA1NPC1RAB9A
SCHEMBL6883428 0.91 ADORA2A (1.00) ADORA2A
SCHEMBL12923671 0.91 ADORA2A (1.00) ADORA2A
SCHEMBL990513 0.91 ADORA2A (1.00) ADORA2A
SCHEMBL991077 0.87 ADORA2A (0.81) ADORA2A
SCHEMBL990483 0.86 ADORA2A (0.75) ADORA2A
SCHEMBL18269264 0.86 ADORA2A (0.75) ADORA2A
SCHEMBL990485 0.86 ADORA2A (0.75) ADORA2A
SCHEMBL6876823 0.84 ADORA2A (0.71) ADORA2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689790-B2 8-AMINO-6-AMIDO-SUBSTITUTED-(1,2,4)TRIAZOLO(1,5-A)PYRIDINES; ADENOSINE RECEPTOR MODULATERS HOFFMANN-LA ROCHE INC. 2004-02-10 US disclosed