SCHEMBL6885776

SCHEMBL6885776

Cc1c(C(O)CC(=O)O)ncn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
PTGDR2 Q9Y5Y4 5/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
GABBR2 O75899 1/20 0.32
GABBR1 Q9UBS5 1/20 0.32
CTSA P10619 1/20 0.32
KDM4E B2RXH2 2/20 0.31
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
CHRM3 P20309 1/20 0.30
MAPT P10636 2/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
GLA P06280 1/20 0.30
STAT1 P42224 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL312703 0.87 TSHR (0.38) CHRM2CHRM1CHRM3ALDH1A1
SCHEMBL12907335 0.80 CYP11B1 (0.37) CYP2C19HIF1ACYP11B1CYP11B2CHRM2
SCHEMBL7377819 0.75 CYP11B1 (0.37) CYP2C19HIF1ACYP11B1CYP11B2CHRM2
SCHEMBL9588293 0.74 CYP11B1 (0.34) CYP11B1CYP11B2
SCHEMBL7534704 0.72 HIF1A (0.37) CYP2C19HIF1APTGDR2KDM4EALDH1A1
SCHEMBL923644 0.72 LMNA (0.37) CYP11B1CYP11B2KDM4EMAPTALDH1A1
SCHEMBL14197521 0.71 KDM4C (0.36) ALDH1A1
SCHEMBL1423832 0.71 TSHR (0.44) CYP2C19MAPTALDH1A1HPGD
SCHEMBL1312709 0.70 SIRT2 (0.39) CYP11B1CYP11B2GABBR2GABBR1
SCHEMBL30946779 0.70 BRD4 (0.34) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1471056-A1 PROCESS FOR PRODUCING FUSED IMIDAZOLE COMPOUND, REFORMATSKY REAGENT IN STABLE FORM, AND PROCESS FOR PRODUCING THE SAME Takeda Chemical Industries, Ltd. (JP) 2004-10-27 EP disclosed