SCHEMBL6887162

SCHEMBL6887162

CN(C)C(=O)C1CCCN1C(=O)c1cc(N)c2nc(-c3ccccc3)nn2c1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.53
USP19 O94966 1/20 0.39
NTRK1 P04629 1/20 0.37
HSD11B1 P28845 1/20 0.37
AVPR2 P30518 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12923690 1.00 ADORA2A (0.53) ADORA2AUSP19NTRK1HSD11B1AVPR2
SCHEMBL6886980 0.86 ADORA2A (0.69) ADORA2A
SCHEMBL6877097 0.83 ADORA2A (0.69) ADORA2A
SCHEMBL12923689 0.82 ADORA2A (0.71) ADORA2A
SCHEMBL6876823 0.82 ADORA2A (0.71) ADORA2A
SCHEMBL6885468 0.82 ADORA2A (0.71) ADORA2A
SCHEMBL6885255 0.79 ADORA2A (0.70) ADORA2A
SCHEMBL6886204 0.78 ADORA2A (0.74) ADORA2A
SCHEMBL6886136 0.78 ADORA2A (0.72) ADORA2A
SCHEMBL6885002 0.77 ADORA2A (0.73) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689790-B2 8-AMINO-6-AMIDO-SUBSTITUTED-(1,2,4)TRIAZOLO(1,5-A)PYRIDINES; ADENOSINE RECEPTOR MODULATERS HOFFMANN-LA ROCHE INC. 2004-02-10 US disclosed