SCHEMBL6887971

SCHEMBL6887971

COC(=O)c1cn(C)nc1C(Cl)(Cl)Cl

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
ADCY10 Q96PN6 1/20 0.39
NR4A2 P43354 2/20 0.37
KMT2A Q03164 4/20 0.37
MAPT P10636 2/20 0.37
F2 P00734 2/20 0.37
MEN1 O00255 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 2/20 0.36
BRD4 O60885 1/20 0.36
CNR2 P34972 1/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5720281 0.84 BAZ2B (0.46) GAALMNAKMT2AMEN1NPC1
SCHEMBL6887159 0.83 GAA (0.68) GAALMNAPOLBNR4A2MAPT
SCHEMBL5720264 0.81 POLB (0.41) GAALMNAPOLBKMT2ARAB9A
SCHEMBL27351594 0.77 ADCY10 (0.43) GAALMNAPOLBADCY10NR4A2
SCHEMBL4443917 0.75 CNR2 (0.47) GAAADCY10NR4A2KMT2AMAPT
SCHEMBL841632 0.75 GAA (0.51) GAAPOLBNR4A2KMT2AMAPT
SCHEMBL25409621 0.74 KDM4E (0.43) GAAADCY10NR4A2KMT2AMAPT
SCHEMBL5653038 0.74 GAA (0.42) GAAADCY10NR4A2KMT2AMAPT
SCHEMBL31499306 0.74 GAA (0.42) GAALMNAADCY10NR4A2KMT2A
SCHEMBL23362881 0.74 NR4A2 (0.40) GAALMNAADCY10NR4A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106467492-B preparation method of polyfluoromethyl pyrazole compound, intermediate and preparation method 联化科技(盐城)有限公司 2019-12-17 CN disclosed
CN-100338029-C Method for producing 2-halogenacyl-3-amino-acrylic acid derivatives BAYER AG (DE) 2007-09-19 CN disclosed
CN-1604889-A Method for producing 2-halogenacyl-3-amino-acrylic acid derivatives BAYER AG (DE) 2005-04-06 CN disclosed
US-6706911-B1 REACTING N-SUBSTITUTED 3-AMINOACRYLIC ESTERS WITH HALOALKYLCARBOXYLIC ANHYDRIDES IN PRESENCE OF BASE; PYRAZOLE-4-CARBOXYLIC ACID CHEMICAL INTERMEDIATES; HALOACYLATION BAYER AKTIENGESELLSCHAFT (DE) 2004-03-16 US disclosed