SCHEMBL6889046

SCHEMBL6889046

CNC(=O)c1cc(N2CCN(C(=O)OC(C)(C)C)C(C)C2)ccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 4/20 0.46
NR1H2 P55055 6/20 0.43
NR1H3 Q13133 5/20 0.43
MAPT P10636 4/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
SUV39H2 Q9H5I1 1/20 0.41
HDAC1 Q13547 1/20 0.41
GPR119 Q8TDV5 2/20 0.41
MAP4K4 O95819 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30082698 0.85 SIRT6 (0.53) SIRT6NR1H2NR1H3MAPTALDH1A1
SCHEMBL24794215 0.85 SIRT6 (0.53) SIRT6NR1H2NR1H3MAPTALDH1A1
SCHEMBL30082668 0.85 SIRT6 (0.53) SIRT6NR1H2NR1H3MAPTALDH1A1
SCHEMBL24792933 0.85 SIRT6 (0.53) SIRT6NR1H2NR1H3MAPTALDH1A1
SCHEMBL16825056 0.84 NR1H2 (0.50) NR1H2NR1H3MAPTALDH1A1LMNA
SCHEMBL31104830 0.84 NR1H2 (0.50) NR1H2NR1H3MAPTALDH1A1LMNA
SCHEMBL18186364 0.84 NR1H2 (0.50) NR1H2NR1H3MAPTALDH1A1LMNA
SCHEMBL30426534 0.84 NR1H2 (0.50) NR1H2NR1H3MAPTALDH1A1LMNA
SCHEMBL31105119 0.84 NR1H2 (0.50) NR1H2NR1H3MAPTALDH1A1LMNA
SCHEMBL23044905 0.84 NR1H2 (0.53) SIRT6NR1H2NR1H3MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045258-A1 CONDENSED AZINE - DERIVATIVES FOR THE TREATMENT OF DISEASES RELATED TO THE ACETYLCHOLINE RECEPTOR N.V. ORGANON (NL) 2011-04-21 WO disclosed