SCHEMBL6889407

SCHEMBL6889407

N#Cc1cccc(-c2cn(Cc3ccc4ccccc4c3)cc2C(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
XDH P47989 2/20 0.44
SLC22A12 Q96S37 2/20 0.44
PLK1 P53350 1/20 0.41
MMP12 P39900 1/20 0.40
MMP13 P45452 1/20 0.40
HTT P42858 1/20 0.40
F11 P03951 1/20 0.39
BRS3 P32247 1/20 0.39
CCR2 P41597 1/20 0.39
PIN1 Q13526 1/20 0.38
TBXAS1 P24557 1/20 0.38
EIF4E P06730 1/20 0.38
ADRA1D P25100 1/20 0.38
CFTR P13569 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6170073 0.86 FNTA (0.44) HTTALDH1A1
SCHEMBL6884036 0.83 MCL1 (0.46) XDHSLC22A12MMP12MMP13HTT
SCHEMBL7100618 0.73 POLB (0.44) HTTADRA1DALDH1A1
SCHEMBL6163480 0.72 POLB (0.44) HTTADRA1DALDH1A1
SCHEMBL7106932 0.71 POLB (0.44) ALDH1A1
SCHEMBL7101526 0.71 CYP19A1 (0.43) XDHSLC22A12HTTBRS3CCR2
SCHEMBL5085509 0.71 SLC22A12 (0.61) XDHSLC22A12HTTF11BRS3
SCHEMBL6165250 0.70 FNTA (0.51) ALDH1A1
SCHEMBL15486418 0.69 ELANE (0.48) XDHCCR2
SCHEMBL7102321 0.69 POLB (0.43) BRS3ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP claimed
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP disclosed