SCHEMBL6889627

SCHEMBL6889627

Cc1c(-c2ccc(C#N)cc2)c(C)n(Cc2ccc(C#N)cc2)c1Cc1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.67
PDE9A O76083 1/20 0.45
PDE1C Q14123 1/20 0.45
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 1/20 0.40
CYP11B1 P15538 2/20 0.40
CYP11B2 P19099 2/20 0.40
CXCR2 P25025 1/20 0.39
CYP19A1 P11511 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6469486 0.83 AR (0.56) ARCYP11B1CYP11B2CYP19A1PTGDR2
SCHEMBL6889022 0.81 AR (0.68) ARCYP11B1CYP11B2CYP19A1PTGDR2
SCHEMBL6466939 0.76 AR (0.67) ARPTGDR2SMN1; SMN2LMNA
SCHEMBL6468889 0.76 AR (0.86) ARPDE9APDE1CALDH1A1CYP11B1
SCHEMBL6469698 0.75 AR (0.61) ARKDM4EPTGDR2LMNA
SCHEMBL24414502 0.75 AR (0.80) ARPDE9APDE1CALDH1A1CYP11B1
SCHEMBL6466328 0.73 AR (0.57) ARALDH1A1CYP11B1CYP11B2KDM4E
SCHEMBL6466315 0.72 AR (0.59) ARALDH1A1CYP11B1CYP11B2CYP19A1
SCHEMBL6468911 0.71 AR (1.00) ARALDH1A1PKMSMN1; SMN2LMNA
SCHEMBL6466727 0.71 AR (0.60) ARALDH1A1CYP11B1CYP11B2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP disclosed