SCHEMBL6889022

SCHEMBL6889022

Cc1c(-c2ccc(C#N)cc2)c(C)n(Cc2ccc(C#N)cc2)c1C

nearest known ligand 0.68

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.68
CYP19A1 P11511 2/20 0.46
CYP11B2 P19099 4/20 0.44
CYP11B1 P15538 3/20 0.44
CCNC P24863 1/20 0.42
CDK8 P49336 1/20 0.42
CYP2A6 P11509 1/20 0.42
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
KLKB1 P03952 1/20 0.39
KLK1 P06870 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468889 0.88 AR (0.86) ARCYP19A1CYP11B2CYP11B1CCNC
SCHEMBL6469486 0.84 AR (0.56) ARCYP19A1CYP11B2CYP11B1CCNC
SCHEMBL24414502 0.84 AR (0.80) ARCYP19A1CYP11B2CYP11B1CCNC
SCHEMBL6466939 0.82 AR (0.67) ARTSHRPTGDR2KLKB1KLK1
SCHEMBL21996432 0.81 AR (0.76) ARCYP19A1CYP11B2CYP11B1LOXL2
SCHEMBL24411064 0.81 AR (0.76) ARCYP19A1CYP11B2CYP11B1CCNC
SCHEMBL24411088 0.81 AR (0.76) ARCYP19A1CYP11B2CYP11B1CCNC
SCHEMBL6889627 0.81 AR (0.67) ARCYP19A1CYP11B2CYP11B1PTGDR2
SCHEMBL6466315 0.81 AR (0.59) ARCYP19A1CYP11B2CYP11B1TSHR
SCHEMBL6884237 0.81 AR (0.57) ARCYP19A1CYP11B2CYP11B1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP disclosed