SCHEMBL6891263

SCHEMBL6891263

CCc1cccc(-c2cccc(C3(C4CCN(C(C)=O)CC4)N=C(C)C(N)=N3)c2)c1

nearest known ligand 0.74

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.74
KCNH2 Q12809 5/20 0.51
BACE2 Q9Y5Z0 3/20 0.51
MAP3K7 O43318 2/20 0.36
TAB1 Q15750 2/20 0.36
PIK3CA P42336 1/20 0.35
GRIN2B Q13224 1/20 0.35
WNT3A P56704 1/20 0.35
BCL2 P10415 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6891914 0.82 BACE1 (0.71) BACE1KCNH2BACE2
SCHEMBL932073 0.74 BACE1 (0.59) BACE1KCNH2BACE2
SCHEMBL6891103 0.70 BACE1 (0.56) BACE1KCNH2BACE2
SCHEMBL6892665 0.69 BACE1 (0.80) BACE1KCNH2BACE2
SCHEMBL4707325 0.68 BACE1 (0.65) BACE1BACE2
SCHEMBL6894615 0.68 BACE1 (0.73) BACE1KCNH2BACE2
SCHEMBL943175 0.68 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL931835 0.68 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL13649187 0.66 HRH3 (0.60) BCL2
SCHEMBL932581 0.66 BACE1 (0.92) BACE1KCNH2BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed