SCHEMBL6892549

SCHEMBL6892549

Cn1c(=O)n(CC(C)(C)CC(F)(F)F)c2ccc(N3CC4CCC3CN4C(=O)OC(C)(C)C)nc21

nearest known ligand 0.81

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 16/20 0.81
CYP3A4 P08684 1/20 0.57
HDAC1 Q13547 2/20 0.42
PARP1 P09874 1/20 0.40
GPR119 Q8TDV5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1502959 0.90 GRM2 (1.00) GRM2CYP3A4HDAC1PARP1
SCHEMBL6894402 0.84 GRM2 (0.77) GRM2CYP3A4HDAC1PARP1GPR119
SCHEMBL6891655 0.84 GRM2 (0.76) GRM2CYP3A4HDAC1PARP1GPR119
SCHEMBL6893813 0.83 GRM2 (0.83) GRM2CYP3A4
SCHEMBL6890927 0.83 GRM2 (0.75) GRM2CYP3A4HDAC1PARP1GPR119
SCHEMBL6890267 0.83 GRM2 (0.86) GRM2CYP3A4HDAC1PARP1
SCHEMBL6894419 0.81 GRM2 (0.83) GRM2CYP3A4
SCHEMBL6889485 0.80 GRM2 (0.78) GRM2CYP3A4
SCHEMBL6892264 0.79 GRM2 (0.79) GRM2CYP3A4
SCHEMBL6893529 0.79 GRM2 (0.80) GRM2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011034741-A1 IMIDAZOPYRIDIN-2-ONE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2011-03-24 WO disclosed