SCHEMBL6894187

SCHEMBL6894187

Cc1ccc(-c2c(C)ncnc2N2CCC(CN)CC2)cn1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 3/20 0.50
GSK3B P49841 1/20 0.50
CHEK1 O14757 1/20 0.46
CHEK2 O96017 1/20 0.46
PIK3CA P42336 7/20 0.45
MTOR P42345 7/20 0.45
RPS6KB1 P23443 3/20 0.43
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
KIT P10721 2/20 0.41
AKT1 P31749 1/20 0.41
CHRM4 P08173 2/20 0.40
PTPN11 Q06124 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10197838 0.79 PIK3CA (0.66) PIK3CAMTORRPS6KB1AKT1
SCHEMBL10196526 0.78 MTOR (0.68) PIK3CAMTOR
SCHEMBL10195779 0.77 PIK3CA (0.68) PIK3CAMTOR
SCHEMBL10195404 0.77 PIK3CA (0.67) PIK3CAMTORRPS6KB1AKT1CHRM4
SCHEMBL6896339 0.76 PIK3CA (0.55) PIK3CAMTOR
SCHEMBL10195993 0.76 PIK3CA (0.64) GSK3BCHEK1CHEK2PIK3CAMTOR
SCHEMBL24632524 0.75 AKT2 (0.44) AKT2GSK3BCHEK1CHEK2PIK3CA
SCHEMBL31625156 0.75 AKT2 (0.44) AKT2GSK3BCHEK1CHEK2PIK3CA
SCHEMBL10197912 0.74 PIK3CA (0.66) PIK3CAMTORCHRM4
SCHEMBL10198433 0.74 PIK3CA (0.70) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092197-A1 5-ALKYNYL PYRIMIDINES AND THEIR USE AS KINASE INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-04 WO disclosed