SCHEMBL6895013

SCHEMBL6895013

CC(=O)c1nc(S(C)(=O)=O)c2sc(C3=C(C(=O)O)N4C(=O)[C@H]([C@@H](C)O)[C@@H]4C3C)cn12

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.34
ESR1 P03372 1/20 0.31
PTGS1 P23219 1/20 0.31
PDE4A P27815 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6886789 1.00 CACNA1C (0.34) CACNA1CESR1PTGS1PDE4A
SCHEMBL7730547 0.92 ABCC2 (0.31)
SCHEMBL7730662 0.92 ABCC2 (0.31)
SCHEMBL6887322 0.89 CACNA1C (0.35) CACNA1CESR1PTGS1PDE4A
SCHEMBL6894605 0.89 CACNA1C (0.35) CACNA1CESR1PTGS1PDE4A
SCHEMBL6887107 0.89 CACNA1C (0.35) CACNA1CESR1PTGS1PDE4A
SCHEMBL6887444 0.85 CACNA1C (0.33) CACNA1CESR1PTGS1PDE4A
SCHEMBL6886997 0.85 ESR1 (0.33) CACNA1CESR1PTGS1PDE4A
SCHEMBL7722383 0.82 PLCG1 (0.34)
SCHEMBL7729826 0.82 ABCC2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677331-B2 HAVING SUBSTITUTED IMIDAZO(5,1-B)THIAZOLE GROUP AT 2-POSITION; MICROBIOCIDES AGAINST BETA-LACTAMASE PRODUCING BACTERIA AND RESISTANT PSEUDOMONAS MEIJI SEIKA KAISHA, LTD. (JP) 2004-01-13 US disclosed