SCHEMBL6900554

SCHEMBL6900554

COc1ccc(COc2cn(-c3ccccc3)c(C=O)cc2=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
ABCB1 P08183 2/20 0.43
GRM5 P41594 1/20 0.43
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
HDAC8 Q9BY41 2/20 0.40
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
BCHE P06276 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LTA4H P09960 1/20 0.39
KCNH2 Q12809 1/20 0.39
MCHR1 Q99705 1/20 0.39
PLA2G4A P47712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2467784 0.88 NPC1 (0.45) ALDH1A1NPC1RAB9ATDP1ABCB1
SCHEMBL12968953 0.83 NPC1 (0.47) ALDH1A1NPC1RAB9ATDP1ABCB1
SCHEMBL9369728 0.82 NPC1 (0.46) ALDH1A1NPC1RAB9ATDP1ABCB1
SCHEMBL9367318 0.81 NPC1 (0.42) NPC1RAB9ATDP1ABCB1GRM5
SCHEMBL9354172 0.81 NPC1 (0.45) ALDH1A1NPC1RAB9ATDP1ABCB1
SCHEMBL9366519 0.81 NPC1 (0.45) NPC1RAB9ATDP1HDAC8MEN1
SCHEMBL2465928 0.80 COMT (0.42) NPC1RAB9AGRM5
SCHEMBL2464192 0.76 COMT (0.54) ABCB1GRM5CTSLCTSB
SCHEMBL9366595 0.73 CSF1R (0.45) ALDH1A1NPC1RAB9ATDP1CTSL
SCHEMBL14124878 0.73 L3MBTL1 (0.41) ALDH1A1NPC1RAB9ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed