SCHEMBL6900641

SCHEMBL6900641

CNC(=O)c1cc(NC(=O)O)cn1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 2/20 0.40
HRAS P01112 1/20 0.40
ESR1 P03372 1/20 0.40
ESR2 Q92731 1/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
HIF1A Q16665 1/20 0.40
P2RY12 Q9H244 1/20 0.39
AR P10275 1/20 0.38
BAZ2B Q9UIF8 1/20 0.38
HPSE Q9Y251 2/20 0.36
NR4A2 P43354 1/20 0.35
TP53 P04637 2/20 0.35
THRB P10828 2/20 0.34
BRD4 O60885 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14535121 0.85 TOP1 (0.45) TOP1HRASESR1ESR2MAPT
SCHEMBL8889890 0.84 TDP1 (0.41) TOP1HRASESR1ESR2MAPT
SCHEMBL24063140 0.83 TOP1 (0.44) TOP1HRASESR1ESR2MAPT
SCHEMBL14002824 0.81 HRAS (0.45) TOP1HRASESR1ESR2MAPT
SCHEMBL6576431 0.81 AR (0.39) TOP1HRASESR1ESR2MAPT
SCHEMBL20581230 0.80 HRAS (0.42) TOP1HRASESR1ESR2MAPT
SCHEMBL5748171 0.80 HRAS (0.42) TOP1HRASESR1ESR2MAPT
SCHEMBL5748174 0.80 TOP1 (0.62) TOP1HRASESR1ESR2MAPT
SCHEMBL14002822 0.80 TOP1 (0.62) TOP1HRASESR1ESR2MAPT
SCHEMBL14509989 0.79 MEN1 (0.49) KDM4EP2RY12TP53SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430028-A2 AROMATIC AND HETEROAROMATIC ACID HALIDES FOR SYNTHESIZING POLYAMIDES Pharmacia Corporation (US) 2004-06-23 EP disclosed
WO-2003018552-A2 AROMATIC AND HETEROAROMATIC ACID HALIDES FOR SYNTHESIZING POLYAMIDES PHARMACIA CORPORATION (US) 2003-03-06 WO disclosed