SCHEMBL6576431

SCHEMBL6576431

Cn1cc(NC(=O)O)cc1C(=O)Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.39
TOP1 P11387 2/20 0.36
HRAS P01112 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
POLB P06746 3/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
HIF1A Q16665 1/20 0.35
P2RY12 Q9H244 1/20 0.35
KMT2A Q03164 4/20 0.34
RAB9A P51151 3/20 0.34
MEN1 O00255 3/20 0.34
HDAC8 Q9BY41 1/20 0.33
NPC1 O15118 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
PKM P14618 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8889890 0.85 TDP1 (0.41) ARTOP1HRASESR1ESR2
SCHEMBL7116896 0.81 POLB (0.35) ARTOP1HRASESR1ESR2
SCHEMBL6900641 0.81 TOP1 (0.40) ARTOP1HRASESR1ESR2
SCHEMBL14535121 0.79 TOP1 (0.45) ARTOP1HRASESR1ESR2
SCHEMBL6527019 0.79 POLB (0.34) ARTOP1HRASESR1ESR2
SCHEMBL4850168 0.77 HRAS (0.49) ARTOP1HRASESR1ESR2
SCHEMBL20581230 0.74 HRAS (0.42) ARTOP1HRASESR1ESR2
SCHEMBL14509989 0.73 MEN1 (0.49) KDM4EP2RY12KMT2ARAB9AMEN1
SCHEMBL3357113 0.73 HSD17B10 (0.44) ARPOLBMAPTKMT2ARAB9A
SCHEMBL20581148 0.71 P2RY12 (0.43) ARTOP1HRASESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1430028-A2 AROMATIC AND HETEROAROMATIC ACID HALIDES FOR SYNTHESIZING POLYAMIDES Pharmacia Corporation (US) 2004-06-23 EP disclosed
EP-1421056-A1 (ALPHA)-HALOENAMINE REAGENTS Pharmacia Corporation (US) 2004-05-26 EP disclosed
WO-2003020684-A1 (ALPHA)-HALOENAMINE REAGENTS PHARMACIA CORPORATION (US) 2003-03-13 WO disclosed
WO-2003018552-A2 AROMATIC AND HETEROAROMATIC ACID HALIDES FOR SYNTHESIZING POLYAMIDES PHARMACIA CORPORATION (US) 2003-03-06 WO disclosed