SCHEMBL6901886

SCHEMBL6901886

O=Nc1cn(-c2cccc(-c3ccccc3)c2)c(CO)c(Br)c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
COMT P21964 13/20 0.47
TET2 Q6N021 1/20 0.37
TET1 Q8NFU7 1/20 0.37
ALDH1A1 P00352 2/20 0.37
FAAH O00519 1/20 0.37
HSP90AA1 P07900 1/20 0.37
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
ATM Q13315 1/20 0.37
MGLL Q99685 1/20 0.37
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
CDK1 P06493 1/20 0.33
SRC P12931 1/20 0.33
ABL2 P42684 1/20 0.33
USP2 O75604 1/20 0.32
CYP1A2 P05177 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14816337 0.84 COMT (0.60) COMTTET2TET1ALDH1A1FAAH
SCHEMBL6900202 0.72 COMT (0.60) COMTTET2TET1ALDH1A1FAAH
SCHEMBL22878779 0.68 COMT (0.43) COMTALDH1A1MAPT
SCHEMBL22878810 0.64 COMT (0.65) COMTTET2TET1ALDH1A1FAAH
SCHEMBL27551731 0.60 FAAH (0.55) COMTTET2TET1ALDH1A1FAAH
SCHEMBL22878794 0.60 COMT (0.59) COMTTET2TET1ALDH1A1HTT
SCHEMBL2467409 0.60 COMT (1.00) COMTALDH1A1FAAHHSP90AA1PKM
SCHEMBL6900205 0.58 COMT (0.78) COMT
SCHEMBL2465251 0.58 COMT (1.00) COMT
SCHEMBL2432898 0.58 COMT (0.74) COMTTET2TET1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed