SCHEMBL6911074

SCHEMBL6911074

CCS(=O)(=O)Nc1nc(-c2ccc(F)cc2C)c2ccc(=O)n(C(C)C)c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 5/20 0.39
RORC P51449 1/20 0.38
CREBBP Q92793 3/20 0.36
GRIN1 Q05586 3/20 0.33
GRIN2B Q13224 3/20 0.33
KMO O15229 1/20 0.33
MAPK8 P45983 1/20 0.33
HMGCR P04035 1/20 0.33
KIT P10721 1/20 0.33
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
TYK2 P29597 1/20 0.32
JAK3 P52333 1/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
CCND2 P30279 1/20 0.32
CCND3 P30281 1/20 0.32
MAP2K4 P45985 1/20 0.32
MAPK13 O15264 1/20 0.32
MAPK12 P53778 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1067521 0.90 RORC (0.36) BRD4RORCMAPK8CDK4CCND1
SCHEMBL1065266 0.83 MAPK14 (0.39) RORCGRIN1GRIN2BMAPK8HMGCR
SCHEMBL1059261 0.83 CDK5 (0.39) RORCGRIN1GRIN2BMAPK8
SCHEMBL1059149 0.81 BRD4 (0.36) BRD4RORCGRIN1GRIN2BHMGCR
SCHEMBL1063029 0.78 HSP90AB1 (0.46) RORCHMGCRMAPK13MAPK12MAPK11
SCHEMBL1063010 0.78 HMGCR (0.37) RORCHMGCRMAPK13MAPK12MAPK11
SCHEMBL1061554 0.77 CCNT1 (0.38) GRIN1GRIN2BCDK4CCND1CCND2
SCHEMBL12122428 0.76 CDK4 (0.34) BRD4RORCGRIN1GRIN2BCDK4
SCHEMBL1065461 0.76 CDK4 (0.34) BRD4RORCGRIN1GRIN2BCDK4
SCHEMBL1064579 0.73 CDK4 (0.42) MAPK8CDK4CCND1CCND2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116697-A1 Novel compounds GLAXOSMITHKLINE LLC 2004-06-17 US claimed