SCHEMBL6915112

SCHEMBL6915112

CC1(C[C@@H](N)C(=O)NC(=O)C2C[C@@H](F)CN2Cc2c(-n3cncn3)ccc(Cl)c2F)CC1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.33
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6922395 0.99 AAK1 (0.32) AAK1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6919094 0.86
SCHEMBL6919199 0.86 F2 (0.39) AAK1
SCHEMBL6919210 0.86 F2 (0.39) AAK1
SCHEMBL6915116 0.81 CFD (0.41)
Hydrochloric Acid SCHEMBL6922397 0.81 CFD (0.40)
Hydrochloric Acid SCHEMBL6916621 0.79 MAOB (0.41) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL6919761 0.78 F2 (0.40) AAK1
SCHEMBL6919684 0.75 F2 (0.42) AAK1
SCHEMBL6921204 0.74 F2 (0.40) AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO claimed