SCHEMBL6917341

SCHEMBL6917341

O=C(O)CCNC(=O)c1ccc(C(=O)C(CC(=O)C2=COC=C(C3=CC=CC(F)(F)C3(F)F)O2)c2ccc(C3CCCCC3)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GCGR P47871 11/20 0.35
CYP2D6 P10635 1/20 0.33
EPHX2 P34913 1/20 0.31
GLP1R P43220 2/20 0.30
PPARD Q03181 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRK1 P41145 1/20 0.30
GCG P01275 3/20 0.30
GIPR P48546 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2647808 0.87 GCGR (0.38) GCGRGCG
SCHEMBL6914041 0.82 GCGR (0.36) GCGRCYP2D6EPHX2PPARDGIPR
SCHEMBL2653731 0.77 HAO1 (0.46) GCGRCYP2D6EPHX2PPARD
SCHEMBL6755519 0.76 GCGR (0.55) GCGRGLP1ROPRM1OPRK1GIPR
SCHEMBL6917335 0.74 DHODH (0.39) GCGRCYP2D6EPHX2GLP1RPPARD
SCHEMBL2654474 0.73 HAO1 (0.42) GCGRCYP2D6EPHX2PPARD
SCHEMBL2647125 0.73 CYP2D6 (0.45) GCGRCYP2D6GLP1ROPRM1OPRK1
SCHEMBL2660182 0.73 GCGR (0.45) GCGRCYP2D6OPRM1OPRK1GCG
SCHEMBL2647568 0.73 GCGR (0.45) GCGRCYP2D6OPRM1OPRK1GCG
SCHEMBL2647399 0.72 PPARD (0.47) GCGRGLP1RPPARDGCGGIPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6762318-B2 CARBOXYLIC ACID OR TETRAZOLE DERIVATIZED SECONDARY AMIDES; ORAL ADMINISTRATION NOVO NORDISK A/S (DK) 2004-07-13 US disclosed
US-20030236292-A1 Stimulant releasing glucose from liver cells; antidiabetic agents PFIZER INC 2003-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236292-A1 Stimulant releasing glucose from liver cells; antidiabetic agents GPR119, GLP1R, GIPR GCGR 4/4885CYP2D6 2704/4885EPHX2 4354/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.