SCHEMBL6917705

SCHEMBL6917705

Nc1nc(-c2cc(-c3ccc(Cl)c(Cl)c3)ncn2)no1

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMO O15229 12/20 0.60
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
NOTUM Q6P988 1/20 0.41
CASP3 P42574 1/20 0.40
DHFR P00374 1/20 0.38
DYRK1A Q13627 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6918443 0.87 KMO (0.65) KMONPC1RAB9ATP53MAPT
SCHEMBL2280592 0.83 KMO (0.60) KMONPC1RAB9ATP53MAPT
SCHEMBL2278992 0.80 KMO (0.56) KMONPC1RAB9ATP53MAPT
SCHEMBL2280622 0.80 KMO (0.56) KMONPC1RAB9ATP53MAPT
SCHEMBL2291147 0.75 KMO (1.00) KMONPC1RAB9ATP53MAPT
SCHEMBL2281232 0.75 KMO (0.51) KMONPC1RAB9ATP53MAPT
SCHEMBL2286344 0.75 KMO (0.51) KMONPC1RAB9ATP53MAPT
SCHEMBL14742330 0.74 KMO (1.00) KMONPC1RAB9AMAPTL3MBTL1
SCHEMBL2227125 0.70 KMO (0.68) KMO
SCHEMBL2229377 0.70 KMO (0.63) KMODYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011091153-A1 CERTAIN KYNURENINE-3-MONOOXYGENASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF CHDI, INC. (US) 2011-07-28 WO disclosed