SCHEMBL6918586

SCHEMBL6918586

CC1(C[C@@H](N)C(=O)NC(=O)[C@@H]2CC(F)(F)CN2Cc2cc(Cl)ccc2-n2cnnn2)CC1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MASP2 O00187 1/20 0.40
F2 P00734 12/20 0.39
PRSS1 P07477 2/20 0.39
F9 P00740 1/20 0.39
F10 P00742 1/20 0.39
PLAT P00750 1/20 0.39
F11 P03951 1/20 0.39
KLKB1 P03952 1/20 0.39
F7 P08709 1/20 0.39
TBXA2R P21731 1/20 0.39
PRSS3 P35030 1/20 0.39
CYP3A4 P08684 5/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
KCNH2 Q12809 3/20 0.36
F12 P00748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6919166 0.89 CYP3A4 (0.41) MASP2F2PRSS1F9F10
SCHEMBL6918798 0.88 F2 (0.39) F2PRSS1F10PLATPRSS3
SCHEMBL6921701 0.81 GPBAR1 (0.45) MASP2F2PRSS1F9F10
SCHEMBL6918584 0.81 F2 (0.50) MASP2F2PRSS1F9F10
SCHEMBL6918590 0.81 F2 (0.50) MASP2F2PRSS1F9F10
SCHEMBL6919210 0.75 F2 (0.39) F2PRSS1F10PLATPRSS3
SCHEMBL6919199 0.75 F2 (0.39) F2PRSS1F10PLATPRSS3
SCHEMBL6918997 0.75 CYP3A4 (0.45) MASP2F2PRSS1F9F10
SCHEMBL6919934 0.75 CYP3A4 (0.45) MASP2F2PRSS1F9F10
SCHEMBL6916861 0.75 CYP3A4 (0.45) MASP2F2PRSS1F9F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO claimed
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO disclosed