SCHEMBL6920108

SCHEMBL6920108

COc1cnc(C(=O)Nc2ccc(F)c([C@]34CO[C@H](C)[C@H]3C(=O)N(C)C(NC(=O)OC(C)(C)C)=N4)c2)cn1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.52
BACE2 Q9Y5Z0 7/20 0.52
CYP2D6 P10635 1/20 0.50
CTSD P07339 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8516737 0.91 BACE1 (0.55) BACE1BACE2CYP2D6CTSD
SCHEMBL11918196 0.87 BACE1 (0.59) BACE1BACE2CYP2D6CTSD
SCHEMBL990426 0.87 BACE1 (0.63) BACE1BACE2CYP2D6
SCHEMBL990541 0.85 BACE1 (0.51) BACE1BACE2CYP2D6
SCHEMBL6921600 0.83 BACE1 (0.53) BACE1BACE2
SCHEMBL6920129 0.81 BACE1 (0.41) BACE1BACE2
SCHEMBL15835731 0.81 BACE1 (0.60) BACE1BACE2CYP2D6CTSD
SCHEMBL990605 0.81 BACE1 (0.61) BACE1BACE2CYP2D6
SCHEMBL6919726 0.80 BACE1 (0.37) BACE1BACE2CTSD
SCHEMBL990549 0.80 BACE1 (0.57) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139594-B2 Fused aminodihydropyrimidone derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2015-09-22 US disclosed
WO-2011009897-A1 FUSED AMINODIHYDROPYRIMIDONE DERIVATIVES EISAI R&D MANAGEMENT CO., LTD (JP) 2011-01-27 WO disclosed