SCHEMBL990541

SCHEMBL990541

COc1cnc(C(=O)Nc2ccc(F)c([C@]34CO[C@H](C)[C@H]3C(=O)N(C)C(N(C(=O)O)C(C)(C)C)=N4)c2)cn1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.51
BACE2 Q9Y5Z0 6/20 0.51
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8516737 0.86 BACE1 (0.55) BACE1BACE2CYP2D6
SCHEMBL990426 0.86 BACE1 (0.63) BACE1BACE2CYP2D6
SCHEMBL6920108 0.85 BACE1 (0.52) BACE1BACE2CYP2D6
SCHEMBL991255 0.83 BACE1 (0.54) BACE1BACE2
SCHEMBL8515016 0.83 BACE1 (0.55) BACE1BACE2
SCHEMBL990549 0.82 BACE1 (0.57) BACE1BACE2
SCHEMBL990605 0.80 BACE1 (0.61) BACE1BACE2CYP2D6
SCHEMBL11913736 0.79 BACE1 (0.60) BACE1BACE2
SCHEMBL991283 0.79 BACE1 (0.42) BACE1BACE2
SCHEMBL990539 0.78 BACE1 (0.37) BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009897-A1 FUSED AMINODIHYDROPYRIMIDONE DERIVATIVES EISAI R&D MANAGEMENT CO., LTD (JP) 2011-01-27 WO disclosed