SCHEMBL692081

SCHEMBL692081

c1ccc(CC[N+]23CCC(CC2)CC3)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 10/20 0.50
BCHE P06276 1/20 0.47
ACHE P22303 1/20 0.47
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA7 P36544 1/20 0.45
CHRNA4 P43681 1/20 0.45
CHRNA10 Q9GZZ6 1/20 0.45
CHRNA9 Q9UGM1 1/20 0.45
CHRM2 P08172 7/20 0.43
CHRM1 P11229 6/20 0.42
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19884914 0.89 CHRM3 (0.46) CHRM3BCHEACHECHRNB2CHRNB4
SCHEMBL10005292 0.85 CHRM3 (0.58) CHRM3
Bromide SCHEMBL14937409 0.83 CHRM3 (0.59) CHRM3CHRM2CHRM1
SCHEMBL2344944 0.79 BCHE (0.65) CHRM3BCHEACHECHRNB2CHRNB4
Bromide SCHEMBL6889492 0.78 BCHE (0.68) CHRM3BCHEACHECHRNB2CHRNB4
Water SCHEMBL31012149 0.78 BCHE (0.62) CHRM3BCHEACHECHRNB2CHRNB4
Hydrochloric Acid SCHEMBL27524696 0.78 BCHE (0.62) CHRM3BCHEACHECHRNB2CHRNB4
SCHEMBL6830020 0.77 CHKA (0.47) HRH3
Bromide SCHEMBL14165975 0.75 CHRM3 (0.56) CHRM3CHRNB2CHRNB4CHRNA3CHRNA7
Bromide SCHEMBL158788 0.71 CHRNB2 (0.71) CHRM3CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2421518-A2 AGGLOMERATE FORMULATIONS INCLUDING ACTIVE PHARMACEUTICAL AGENTS WITH TARGETED PARTICLE SIZES Schering Corporation (US) 2012-02-29 EP disclosed
WO-2010124203-A2 AGGLOMERATE FORMULATIONS INCLUDING ACTIVE PHARMACEUTICAL AGENTS WITH TARGETED PARTICLE SIZES SCHERING CORPORATION (US) 2010-10-28 WO disclosed
EP-2119716-A1 AZA-BRIDGED-RING COMPOUND Astellas Pharma Inc. (JP) 2009-11-18 EP disclosed
EP-1442027-A1 SUBSTITUTED DIPHENYLOXAZOLES, THE SYNTHESIS THEREOF, AND THE USE THEREOF AS FLUORESCENCE PROBES 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2004-08-04 EP disclosed
WO-2003031419-A1 SUBSTITUTED DIPHENYLOXAZOLES, THE SYNTHESIS THEREOF, AND THE USE THEREOF AS FLUORESCENCE PROBES 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2003-04-17 WO disclosed