SCHEMBL6922716

SCHEMBL6922716

Cc1cc(C#N)c2c3ncnc(Cl)c3n(C)c2n1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 3/20 0.51
CRHR1 P34998 5/20 0.34
KDM5A P29375 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP3A4 P08684 1/20 0.33
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6924927 0.79 ABCC1 (0.48) ABCC1KDM4ELRRK2
SCHEMBL14752628 0.65 MEN1 (0.43) KDM5AALDH1A1KDM4EGLAHPGD
SCHEMBL3484040 0.61 PSMB8 (0.36) LRRK2
SCHEMBL21120068 0.60 KDM5A (0.40) KDM5AALDH1A1KDM4EGLAHPGD
SCHEMBL6923654 0.60 ABCC1 (0.48) ABCC1ALDH1A1CYP3A4KDM4EGLA
SCHEMBL17857294 0.60 ALDH1A1 (0.40) CRHR1KDM5AALDH1A1KDM4EGLA
SCHEMBL12365636 0.60 EGLN2 (0.40) ALDH1A1CYP3A4HPGD
SCHEMBL9649994 0.60 KHK (0.44) KDM5AALDH1A1KDM4EHPGDMAPK1
SCHEMBL31507346 0.60 KHK (0.44) KDM5AALDH1A1CYP3A4KDM4EGLA
SCHEMBL6826551 0.58 ABCC1 (0.39) ABCC1ALDH1A1CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed