SCHEMBL6922950

SCHEMBL6922950

CC(C)=CCNc1n[nH]c2cccnc12

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 19/20 0.52
CCNB2 O95067 1/20 0.45
CDK1 P06493 1/20 0.45
CCNB1 P14635 1/20 0.45
CCNB3 Q8WWL7 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923982 0.88 GRM4 (0.49) GRM4
SCHEMBL6923007 0.82 GRM4 (0.53) GRM4
SCHEMBL17011306 0.79 GRM4 (0.59) GRM4
SCHEMBL28939044 0.77 GRM4 (0.57) GRM4
SCHEMBL19801454 0.74 GRM4 (0.63) GRM4
SCHEMBL19100876 0.74 GRM4 (0.61) GRM4
Hydrochloric Acid SCHEMBL30549482 0.69 GRM4 (0.52) GRM4
SCHEMBL6923917 0.69 GRM4 (1.00) GRM4
SCHEMBL6923497 0.68 GRM4 (1.00) GRM4CDK1
SCHEMBL2359725 0.67 GRM4 (1.00) GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011100607-A1 PYRAZOLOPYRIDINE, PYRAZOLOPYRAZINE, PYRAZOLOPYRIMIDINE, PYRAZOLOTHIOPHENE AND PYRAZOLOTHIAZOLE COMPOUNDS AS MGLUR4 ALLOSTERIC POTENTIATORS, COMPOUNDS, AND METHODS OF TREATING NEUROLOGICAL DYSFUNCTION VANDERBILT UNIVERSITY (US) 2011-08-18 WO disclosed