SCHEMBL692578

SCHEMBL692578

C=CC(=O)OC(C=C)OCC(O)O

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.38
ALDH1A1 P00352 3/20 0.32
TP53 P04637 2/20 0.32
HIF1A Q16665 2/20 0.32
CYP3A4 P08684 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL277923 0.79 TSHR (0.39) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL5485731 0.78 TSHR (0.39) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL4563557 0.78 TSHR (0.35) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL11252991 0.78 TSHR (0.35) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL18224490 0.77 TSHR (0.39) TSHRALDH1A1
SCHEMBL14797171 0.74 TSHR (0.37) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL8752829 0.73 TSHR (0.35) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL11247857 0.72 TSHR (0.32) TSHRALDH1A1TP53HIF1ACYP3A4
SCHEMBL6274690 0.72 TSHR (0.49) TSHRALDH1A1CYP3A4
SCHEMBL8752830 0.71 TSHR (0.34) TSHRALDH1A1TP53HIF1ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4214253-A1 ULTRAVIOLET-ABSORBING ACRYLIC COPOLYMER FOR THE PRODUCTION OF FLEXIBLE INTRAOCULAR LENS Acrylian (FR) 2023-07-26 EP claimed
CN-108348642-B Hydrophobic, crosslinked and cinnamyl alcohol-based acrylic copolymers for intraocular lenses 阿库里恩公司 2022-01-28 CN claimed
US-10626206-B2 Acrylic copolymer, which is hydrophobic, cross-linked and based on cinnamic alcohol, for intraocular lenses ACRYLIAN (FR) 2020-04-21 US claimed
EP-3373992-B1 ACRYLIC COPOLYMER, WHICH IS HYDROPHOBIC, CROSS-LINKED AND BASED ON CINNAMIC ALCOHOL, FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2020-04-08 EP claimed
US-20180312619-A1 ACRYLIC COPOLYMER, WHICH IS HYDROPHOBIC, CROSS-LINKED AND BASED ON CINNAMIC ALCOHOL, FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2018-11-01 US claimed
US-9907881-B2 Crosslinked, hydrophobic acrylic copolymer made of 2-phenoxytetraethylene-glycol acrylate and intended for intraocular lenses ACRYLIAN (FR) 2018-03-06 US claimed
EP-3110464-B1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2-PHENOXY-TETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2017-11-01 EP claimed
US-20160331864-A1 CROSSLINKED, HYDROPHOBIC ACRYLIC COPOLYMER MADE OF 2- PHENOXYTETRAETHYLENE-GLYCOL ACRYLATE AND INTENDED FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2016-11-17 US claimed
US-8470034-B2 Hydrophobic acrylic polymer material for an intraocular lens having enhanced flexibility due to the use of a transfer agent ACRYLIAN (FR) 2013-06-25 US claimed
EP-2285427-B1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS, HAVING AN ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT ACRYLIAN (FR) 2012-02-29 EP claimed
US-20110245442-A1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS HAVING ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT CRISTALENS INDUSTRIE (FR) 2011-10-06 US claimed
EP-4214253-A1 ULTRAVIOLET-ABSORBING ACRYLIC COPOLYMER FOR THE PRODUCTION OF FLEXIBLE INTRAOCULAR LENS Acrylian (FR) 2023-07-26 EP disclosed
US-10626206-B2 Acrylic copolymer, which is hydrophobic, cross-linked and based on cinnamic alcohol, for intraocular lenses ACRYLIAN (FR) 2020-04-21 US disclosed
EP-3373992-B1 ACRYLIC COPOLYMER, WHICH IS HYDROPHOBIC, CROSS-LINKED AND BASED ON CINNAMIC ALCOHOL, FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2020-04-08 EP disclosed
US-20180312619-A1 ACRYLIC COPOLYMER, WHICH IS HYDROPHOBIC, CROSS-LINKED AND BASED ON CINNAMIC ALCOHOL, FOR INTRAOCULAR LENSES ACRYLIAN (FR) 2018-11-01 US disclosed
US-8470034-B2 Hydrophobic acrylic polymer material for an intraocular lens having enhanced flexibility due to the use of a transfer agent ACRYLIAN (FR) 2013-06-25 US disclosed
US-20110245442-A1 HYDROPHOBIC ACRYLIC POLYMER MATERIAL FOR AN INTRAOCULAR LENS HAVING ENHANCED FLEXIBILITY DUE TO THE USE OF A TRANSFER AGENT CRISTALENS INDUSTRIE (FR) 2011-10-06 US disclosed