SCHEMBL6928230

SCHEMBL6928230

OC1CCN(c2ccc(-c3nc(-c4ccc(Cl)c(Cl)c4)c[nH]3)cn2)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.45
MCHR1 Q99705 2/20 0.41
MELK Q14680 3/20 0.41
MGLL Q99685 1/20 0.39
MAPK1 P28482 1/20 0.39
PRKAB2 O43741 3/20 0.39
PRKAG1 P54619 3/20 0.39
PRKAA2 P54646 3/20 0.39
PRKAA1 Q13131 3/20 0.39
PRKAG3 Q9UGI9 3/20 0.39
PRKAG2 Q9UGJ0 3/20 0.39
PRKAB1 Q9Y478 3/20 0.39
DGAT1 O75907 2/20 0.39
KCNH2 Q12809 2/20 0.39
ALOX5AP P20292 2/20 0.39
ADK P55263 1/20 0.38
ADORA2A P29274 1/20 0.37
RET P07949 1/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920372 0.95 CNR2 (0.50) CNR2MCHR1MGLLDGAT1KCNH2
SCHEMBL6927037 0.88 ITGB2 (0.42) MAPK1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL6928989 0.87 PIM1 (0.45) CNR2MELKMGLLRET
SCHEMBL6924483 0.85 CNR2 (0.49) CNR2MELKMGLLDGAT1KCNH2
SCHEMBL6925625 0.83 MAP4K4 (0.42) CNR2MGLLDGAT1KCNH2ADORA2A
SCHEMBL6921878 0.82 CNR2 (0.45) CNR2MGLLDGAT1KCNH2ADORA2A
SCHEMBL6927498 0.82 ITGB2 (0.41) CNR2RET
SCHEMBL6920358 0.81 CNR2 (0.52) CNR2MELKMGLLKCNH2RET
SCHEMBL6924929 0.81 CNR2 (0.39) CNR2MELKDGAT1KCNH2RET
SCHEMBL6924520 0.80 CNR2 (0.51) CNR2MGLLDGAT1KCNH2RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R CNR2 122/4885MCHR1 61/4885MELK 1367/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.