SCHEMBL6920358

SCHEMBL6920358

Clc1ccc(-c2c[nH]c(-c3ccc(N4CCNCC4)nc3)n2)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.52
RET P07949 3/20 0.46
NMT1 P30419 1/20 0.44
MAP3K11 Q16584 1/20 0.44
ADRB1 P08588 1/20 0.43
MGLL Q99685 1/20 0.42
IL2 P60568 1/20 0.41
MAP4K1 Q92918 1/20 0.41
JAK2 O60674 1/20 0.41
GPR119 Q8TDV5 1/20 0.41
KCNH2 Q12809 1/20 0.41
CACNA1C Q13936 1/20 0.41
ASIC3 Q9UHC3 1/20 0.41
MELK Q14680 1/20 0.41
MAPK7 Q13164 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6929138 0.88 FAAH (0.46) CNR2RETMAP3K11ADRB1IL2
SCHEMBL6924520 0.87 CNR2 (0.51) CNR2RETMGLLIL2MAP4K1
SCHEMBL6927892 0.86 DYRK1A (0.49) NMT1PRKD3PRKD1
SCHEMBL6920372 0.86 CNR2 (0.50) CNR2RETMGLLKCNH2
SCHEMBL6927756 0.85 CNR2 (0.52) CNR2MGLLKCNH2
SCHEMBL6925085 0.85 CNR2 (0.49) CNR2MGLL
SCHEMBL6927450 0.85 CNR2 (0.49) CNR2MGLL
SCHEMBL6924483 0.85 CNR2 (0.49) CNR2RETMGLLKCNH2MELK
SCHEMBL6928035 0.84 CNR2 (0.48) CNR2RETMGLLKCNH2ZAP70
SCHEMBL6927253 0.84 CNR2 (0.48) CNR2RETMGLLKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed
WO-2000066578-A1 COMPOUNDS FOR THE TREATMENT OF OBESITY PFIZER PRODUCTS INC. (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R CNR2 122/4885RET 1562/4885NMT1 566/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.