SCHEMBL6929183

SCHEMBL6929183

Clc1nc[nH]c1CCCN1CC[C@H]2C[C@H](Cc3ccccc3)CC[C@H]21

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.35
CCR3 P51677 4/20 0.34
SIGMAR1 Q99720 2/20 0.34
GRIN2B Q13224 3/20 0.34
GRIN2A Q12879 1/20 0.34
TMEM97 Q5BJF2 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680066 1.00 HRH3 (0.35) HRH3CCR3SIGMAR1GRIN2BGRIN2A
SCHEMBL6931011 0.84 GRIN2B (0.35) HRH3CCR3SIGMAR1GRIN2BGRIN2A
SCHEMBL6925057 0.80 HRH3 (0.53) HRH3
SCHEMBL6930156 0.80 HRH3 (0.53) HRH3
SCHEMBL7066795 0.76 CCR3 (0.37) HRH3CCR3SIGMAR1GRIN2BTMEM97
SCHEMBL7068153 0.74 CCR3 (0.50) CCR3SIGMAR1
SCHEMBL7069134 0.74 CCR3 (0.50) CCR3SIGMAR1
SCHEMBL7068156 0.74 CCR3 (0.50) CCR3SIGMAR1
SCHEMBL7071904 0.74 CCR3 (0.50) CCR3SIGMAR1
SCHEMBL6931066 0.68 TMEM97 (0.49) HRH3SIGMAR1GRIN2BGRIN2ATMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242074-A4 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-01-29 EP claimed
EP-1242074-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-09-25 EP claimed
US-6369076-B1 ANALGESICS MERCK & CO. INC. 2002-04-09 US claimed
WO-2001032171-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO claimed
EP-1242074-A4 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-01-29 EP disclosed
EP-1242074-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-09-25 EP disclosed
US-6369076-B1 ANALGESICS MERCK & CO. INC. 2002-04-09 US disclosed
WO-2001032171-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO disclosed