SCHEMBL7068153

SCHEMBL7068153

c1ccc(C[C@@H]2CC[C@@H]3[C@@H](CCN3Cc3ccccc3)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 1/20 0.50
ALDH1A1 P00352 3/20 0.44
HTR1A P08908 2/20 0.44
ATM Q13315 2/20 0.43
SIGMAR1 Q99720 3/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7069134 1.00 CCR3 (0.50) CCR3ALDH1A1HTR1AATMSIGMAR1
SCHEMBL7068156 1.00 CCR3 (0.50) CCR3ALDH1A1HTR1AATMSIGMAR1
SCHEMBL7071904 1.00 CCR3 (0.50) CCR3ALDH1A1HTR1AATMSIGMAR1
SCHEMBL3176956 0.82 HTR1A (0.51) HTR1ASIGMAR1HTT
SCHEMBL8301747 0.82 HTR1A (0.51) HTR1ASIGMAR1HTT
SCHEMBL7068562 0.80 GRIN2B (0.62) GAAHTT
SCHEMBL7071755 0.80 GRIN2B (0.62) GAAHTT
SCHEMBL6931066 0.76 TMEM97 (0.49) SIGMAR1KDM4E
SCHEMBL7069836 0.76 TMEM97 (0.49) SIGMAR1KDM4E
SCHEMBL7066795 0.76 CCR3 (0.37) CCR3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242074-A4 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-01-29 EP disclosed
EP-1242074-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-09-25 EP disclosed
US-6369076-B1 ANALGESICS MERCK & CO. INC. 2002-04-09 US disclosed
WO-2001032171-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO disclosed