SCHEMBL6929503

SCHEMBL6929503

COC(=O)CCc1[nH]c(Cl)nc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.42
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 2/20 0.40
TSHR P16473 3/20 0.39
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
ALOX12 P18054 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
MAPK1 P28482 2/20 0.36
KAT2B Q92831 2/20 0.36
LCK P06239 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6930989 0.72 EGFR (0.39) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL6929905 0.70 EGFR (0.45) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL31180118 0.66 KDM4E (0.42) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL22307574 0.66 TSHR (0.41) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL5307615 0.63 MAPT (0.54) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL17129771 0.62 TSHR (0.41) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL21679094 0.62 CYP11B1 (0.46) EGFRKDM4EALDH1A1HSD17B10TSHR
SCHEMBL3929708 0.62 KDM4E (0.42) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL23164498 0.61 KDM4E (0.41) EGFRKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL7457649 0.61 HTT (0.48) KDM4EALDH1A1HSD17B10SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242074-A4 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO INC (US) 2003-01-29 EP disclosed
EP-1242074-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS Merck & Co., Inc. (US) 2002-09-25 EP disclosed
US-6369076-B1 ANALGESICS MERCK & CO. INC. 2002-04-09 US disclosed
WO-2001032171-A1 5-BENZYL-OCTAHYDROINDOLE AND 6-BENZYL-DECAHYDROQUINOLINE NMDA/NR2B ANTAGONISTS MERCK & CO., INC. (US) 2001-05-10 WO disclosed