SCHEMBL693019

SCHEMBL693019

CCc1cc(Cc2cc(C)c(N=C=O)c(CC)c2)cc(C)c1N=C=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.47
GABRB2 P47870 2/20 0.47
SHBG P04278 1/20 0.38
CYP3A4 P08684 2/20 0.37
TSHR P16473 1/20 0.37
TRPA1 O75762 1/20 0.33
HMGB1 P09429 1/20 0.33
CXCL12 P48061 1/20 0.33
CYP1A2 P05177 1/20 0.32
DHFR P00374 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28306014 0.91 GABRA1 (0.48) GABRA1GABRB2CYP3A4TSHRTRPA1
SCHEMBL80318 0.89 GABRA1 (0.59) GABRA1GABRB2SHBGCYP3A4TSHR
SCHEMBL28673397 0.88 GABRA1 (0.46) GABRA1GABRB2SHBGCYP3A4TSHR
SCHEMBL940373 0.87 CYP3A4 (0.43) GABRA1GABRB2SHBGCYP3A4TSHR
SCHEMBL27550639 0.81 GABRA1 (0.50) GABRA1GABRB2CYP3A4TRPA1
SCHEMBL28928606 0.81 GABRA1 (0.40) GABRA1GABRB2CYP3A4TSHRTRPA1
SCHEMBL28260919 0.81 GABRA1 (0.50) GABRA1GABRB2CYP3A4TSHRCYP1A2
SCHEMBL15800800 0.79 GABRA1 (0.39) GABRA1GABRB2SHBGCYP3A4TSHR
SCHEMBL13087103 0.79 HMGB1 (0.47) GABRA1GABRB2SHBGCYP3A4TSHR
SCHEMBL17907296 0.79 GABRA1 (0.47) GABRA1GABRB2CYP3A4TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037943-A1 STABILIZED MOLDING COMPOUNDS COMPRISED OF BIOLOGICALLY DEGRADABLE MATERIALS BAYER AG (DE) 2000-09-27 EP claimed
WO-1999029768-A1 STABILIZED MOLDING COMPOUNDS COMPRISED OF BIOLOGICALLY DEGRADABLE MATERIALS BAYER AKTIENGESELLSCHAFT (DE) 1999-06-17 WO claimed
US-11319477-B2 Breaker additives for extended delay in removal of oil-based filter cakes HALLIBURTON ENERGY SERVICES, INC. (US) 2022-05-03 US disclosed
WO-2021076158-A1 BREAKER ADDITIVES FOR EXTENDED DELAY IN REMOVAL OF OIL-BASED FILTER CAKES HALLIBURTON ENERGY SERVICES, INC. (US) 2021-04-22 WO disclosed
US-10478045-B2 Flexible tube for an endoscope, adhesive for an endoscope, endoscope-type medical device, as well as method of producing a flexible tube for an endoscope and method of producing an endoscope-type medical device FUJIFILM CORPORATION (JP) 2019-11-19 US disclosed
EP-3000834-B1 FLEXIBLE TUBE FOR AN ENDOSCOPE, ADHESIVE FOR AN ENDOSCOPE, ENDOSCOPE-TYPE MEDICAL DEVICE, AS WELL AS METHOD OF PRODUCING A FLEXIBLE TUBE FOR AN ENDOSCOPE AND METHOD OF PRODUCING AN ENDOSCOPE-TYPE MEDICAL DEVICE FUJIFILM CORP (JP) 2018-10-24 EP disclosed
US-20160088998-A1 FLEXIBLE TUBE FOR AN ENDOSCOPE, ADHESIVE FOR AN ENDOSCOPE, ENDOSCOPE-TYPE MEDICAL DEVICE, AS WELL AS METHOD OF PRODUCING A FLEXIBLE TUBE FOR AN ENDOSCOPE AND METHOD OF PRODUCING AN ENDOSCOPE-TYPE MEDICAL DEVICE FUJIFILM CORPORATION (JP) 2016-03-31 US disclosed
EP-3000834-A1 FLEXIBLE TUBE FOR AN ENDOSCOPE, ADHESIVE FOR AN ENDOSCOPE, ENDOSCOPE-TYPE MEDICAL DEVICE, AS WELL AS METHOD OF PRODUCING A FLEXIBLE TUBE FOR AN ENDOSCOPE AND METHOD OF PRODUCING AN ENDOSCOPE-TYPE MEDICAL DEVICE Fujifilm Corporation (JP) 2016-03-30 EP disclosed
US-8586507-B2 Oil based drilling fluids with enhanced stability at high temperatures HALLIBURTON ENERGY SERVICES, INC. (US) 2013-11-19 US disclosed
US-20120258893-A1 Oil Based Drilling Fluids With Enhanced Stability at High Temperatures HALLIBURTON ENERGY SERVICES, INC. (US) 2012-10-11 US disclosed
EP-2421931-A1 METHOD FOR ENHANCING STABILITY OF OIL BASED DRILLING FLUIDS AT HIGH TEMPERATURES Halliburton Energy Services, Inc. (US) 2012-02-29 EP disclosed
US-6720403-B1 GOOD WHITENESS RETENTION, HIGH HEAT-SET EFFICIENCY; POLYMERIC GLYCOL, ALKYL SUBSTITUTED METHYLENEBIS(4-ISOCYANATOBENZENE), A DOUBLY-HINDERED DIAMINE E.I. DUPONT DE NEMOURS AND CO. 2004-04-13 US disclosed
EP-1263000-B1 Flat cable FURUKAWA ELECTRIC CO LTD (JP) 2004-03-17 EP disclosed
US-6608256-B2 Flat cable THE FURUKAWA ELECTRIC CO., LTD. (JP) 2003-08-19 US disclosed
US-20030024729-A1 Flat cable FURUKAWA ELECTRIC CO., LTD., THE (JP) 2003-02-06 US disclosed
EP-1263000-A1 Flat cable THE FURUKAWA ELECTRIC CO., LTD. (JP) 2002-12-04 EP disclosed
EP-1037943-A1 STABILIZED MOLDING COMPOUNDS COMPRISED OF BIOLOGICALLY DEGRADABLE MATERIALS BAYER AG (DE) 2000-09-27 EP disclosed
WO-1999029768-A1 STABILIZED MOLDING COMPOUNDS COMPRISED OF BIOLOGICALLY DEGRADABLE MATERIALS BAYER AKTIENGESELLSCHAFT (DE) 1999-06-17 WO disclosed
US-5360888-A Polymeric carbodiimides with polylactams RHEIN CHEMIE RHEINAU GMBH (DE) 1994-11-01 US disclosed
EP-0567884-A1 Hydrolysis-stable polyamides RHEIN CHEMIE RHEINAU GmbH (DE) 1993-11-03 EP disclosed