SCHEMBL6930316

SCHEMBL6930316

C[C@@H](NC(=O)c1cnc(OCc2ccncc2)c(N)c1)C1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 7/20 0.48
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GPR132 Q9UNW8 1/20 0.41
F11 P03951 1/20 0.41
CNR2 P34972 5/20 0.40
IDO1 P14902 1/20 0.40
SMYD3 Q9H7B4 2/20 0.39
WDR5 P61964 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6927899 0.89 CNR1 (0.47) CNR1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL6930244 0.89 CNR1 (0.46) CNR1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL6930900 0.86 CNR1 (0.44) CNR1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL6930980 0.86 CNR1 (0.44) CNR1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL2158694 0.82 GABRA5 (0.51) KDM4EALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL2158698 0.82 GABRA5 (0.51) KDM4EALDH1A1HPGDCYP1A2CYP3A4
SCHEMBL6928005 0.77 GABRA5 (0.51) IDO1
SCHEMBL6930043 0.76 SMYD3 (0.45) CNR1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL6931215 0.75 GRM5 (0.49) CNR1KDM4EALDH1A1HPGDCYP1A2
SCHEMBL6928147 0.74 NOX1 (0.48) CNR1KDM4EALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035324-A1 O-BENZYL NICOTINAMIDE ANALOGS AS MGLUR5 POSITIVE ALLOSTERIC MODULATORS VANDERBILT UNIVERSITY (US) 2011-03-24 WO disclosed