SCHEMBL6930957

SCHEMBL6930957

CC(C)(C)OC(Cn1c(N)nc2ccccc21)C(N)C=O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
POLB P06746 1/20 0.45
CXCR4 P61073 1/20 0.44
F2R P25116 1/20 0.43
TLR8 Q9NR97 3/20 0.43
KCNH2 Q12809 1/20 0.40
NOD1 Q9Y239 4/20 0.40
TNF P01375 2/20 0.40
NOD2 Q9HC29 2/20 0.40
CXCL8 P10145 2/20 0.40
SOS1 Q07889 1/20 0.40
KMT2A Q03164 3/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL6933379 0.99 HTT (0.46) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL989222 0.71 HTT (0.67) HTTCYP1A2CYP2D6POLBCXCR4
Bromide SCHEMBL6932626 0.70 HTT (0.50) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL6930955 0.69 F2R (0.47) HTTCYP1A2CYP2D6POLBCXCR4
Bromide SCHEMBL6933374 0.68 F2R (0.47) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL23319549 0.68 HTT (0.62) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL990194 0.68 HTT (0.67) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL20641347 0.68 HTT (0.62) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL1992429 0.66 CYP1A2 (1.00) HTTCYP1A2CYP2D6POLBCXCR4
SCHEMBL14891383 0.66 HTT (0.63) HTTCYP1A2CYP2D6POLBCXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6660870-B1 Serotonergic compounds which possess agonist activity at 5-HT2 receptors effectively lower and control normal and elevated IOP and are useful for treating glaucoma ALCON, INC. (CH) 2003-12-09 US disclosed